2-[1-[2-Cyclopropyl-1-(2-fluorophenyl)-2-oxoethyl]-4-(Methylthio)-3-piperidinylidene]acetic Acid - Names and Identifiers
2-[1-[2-Cyclopropyl-1-(2-fluorophenyl)-2-oxoethyl]-4-(Methylthio)-3-piperidinylidene]acetic Acid - Physico-chemical Properties
Molecular Formula | C19H22FNO3S
|
Molar Mass | 363.45 |
Storage Condition | 2-8℃ |
2-[1-[2-Cyclopropyl-1-(2-fluorophenyl)-2-oxoethyl]-4-(Methylthio)-3-piperidinylidene]acetic Acid - Introduction
R-106583, also known as Prasugrel metabolite, is a drug compound. It is the main metabolite of Prasugrel, an antiplatelet drug used to prevent cardiovascular events.
The chemical properties of the R-106583 are white crystalline powder. It has low solubility in water, but has good solubility in organic solvents. R-106583 has antiplatelet activity, can effectively inhibit platelet aggregation, and prevent thrombosis.
The main use of R-106583 is as a metabolite of Prasugrel for pharmacokinetic and drug metabolism research. By studying its metabolic process and mechanism of action, we can better understand the pharmacodynamic properties and metabolic pathways of Prasugrel.
Regarding the preparation method, R-106583 is produced by metabolism in the body of Prasugrel. Prasugrel is oxidized to R-106583 in the human body through the catalytic action of cytochrome P450 enzymes.
When using R-106583, you need to pay attention to its safety. Although R-106583 is a metabolite of Prasugrel, it must be handled and used in accordance with chemical safety practices. During use, avoid direct contact with skin, eyes and respiratory tract, and maintain a good ventilation environment. In addition, it also needs to be stored and handled in accordance with relevant regulations.
To sum up, R-106583 is a metabolite of Prasugrel and has anti-platelet activity. It is mainly used in drug metabolism research to better understand the pharmacodynamic properties and metabolic pathways of Prasugrel. Need to pay attention to the use of the need to follow the relevant safety procedures.
Last Update:2024-04-09 21:49:45